somatostatin receptor — TargetMol Chemicals

Cat No.	Product Name	Synonyms	Targets
T2584	Octreotide	SMS 201-995	Somatostatin
	Octreotide (SMS 201-995) is a potent inhibitor of growth hormone, glucagon, and insulin.		Somatostatin
TP2207	Pasireotide Acetate		Somatostatin
	Pasireotide Acetate is a stable cyclohexapeptide somatostatin mimic		Somatostatin
T9692	Paltusotine		Somatostatin
	Paltusotine is a nonpeptide, small molecule somatostatin type 2 (SST2) receptor agonist with high oral bioavailability. Paltusotine maintains GH and IGF-1 levels in acromegaly patients		Somatostatin
T4119	Octreotide Acetate	SMS 201995,Longastatin,Sandostatin,SMS 201-995 (acetate)	Somatostatin
	Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.		Somatostatin
TP2045	CH 275
	Potent somatostatin receptor 1 (sst1) agonist; displays selectivity for sst1 (IC50 values are 30.9 nM, 345 nM, > 1 μM, > 10 μM and > 10μM for human sst1, sst3, sst4, sst2 and sst5 respectively). Attenuates somatostatin r...
T28743	Seglitide acetate	MK 678,MK678,MK-678	Somatostatin
	Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.		Somatostatin
TP2052L	CTOP acetate		Opioid Receptor
	CTOP acetate is a somatostatin analogue and a μ-opioid receptor antagonist.		Opioid Receptor
TP1346	CYN 154806 TFA	CYN 154806 TFA	Somatostatin
	CYN 154806 TFA is a cyclic octapeptide and an effective selective somatostatin sst2 receptor antagonist. For the recombinant sst2, sst1, sst3, sst4 and sst5 receptors, the pIC50 values are 8.58, 5.41, 6.07, 5.76 and 6.48...		Somatostatin
T27787L	L-797,591 hydrochloride	L-797,591 hydrochloride(217480-24-5 Free base)
	L-797,591 hydrochloride is active for somatostatin receptor isoform 1 (SSTR1). L-797,591 hydrochloride is commonly used in combination with AG1478 to enhance p-ERK5 expression in SSTR1 cells. L-797,591 hydrochloride sign...
TP2050L	CTAP(TFA） (103429-32-9 free base)	CTAP(TFA）	Opioid Receptor
	CTAP(TFA) (103429-32-9 free base) is a potent, highly selective, and brain-penetrant antagonist of the μ-opioid receptor with IC50 of 3.5 nM. It displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somato...		Opioid Receptor
T22907	L-817,818		Others
	somatostatin sst5 receptor agonist		Others
T28298	Pasireotide diaspartate	SOM-230,SOM230,trade name: Signifor,SOM 230,Signifor LAR
	Pasireotide is a somatostatin analog with a 40-fold increased affinity to somatostatin receptor 5 compared to other somatostatin analogs.
T23073	NNC 26-9100		Others
	Somatostatin sst4 receptor agonist		Others
T27761	L-054,522	L054,522
	L-054,522 is potent, selective agonists of somatostatin receptor.
T27783	L-779976	L-779,976,L779,976,L779976,L 779976,L 779,976
	L-779,976 is an agonist of somatostatin receptor.
T22487	(1R,1'S,3'R/1R,1'R,3'S)-L-054,264		Others
	somatostatin sst2 receptor agonist		Others
T31606	EE 581	EE581,EE-581
	EE 581 can be used to label the somatostatin receptor.
T24860	TC-G1003	TC G1003
	TC-G1003 is an effective agonist of the somatostatin sst2 receptor.
T27787	L-797,591
	L-797,591 is a selective agonist of somatostatin receptor subtype 1.
T28220	NVP ACQ090	NVP-ACQ090,ACQ090,ACQ 090,NVPACQ090,ACQ-090
	NVP ACQ090 is a potent and subtype-selective somatostatin sst(3) receptor antagonist.